Benzquinamide

{{Short description|Chemical compound}}

{{redirect|Quantril|the surname|Quantrill}}

{{Drugbox

| Verifiedfields = changed

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| verifiedrevid = 459955149

| IUPAC_name = 3-(Diethylcarbamoyl)-9,10-dimethoxy-1H,2H,3H,4H,6H,7H,11bH-pyrido[2,1-a]isoquinolin-2-yl acetate

| image = Benzquinamide.svg

| image_class = skin-invert-image

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| tradename = Promecon, Quantril, Emete-Con

| licence_EU =

| licence_US = Quantril

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| legal_AU =

| legal_BR = C1

| legal_BR_comment = {{Cite web |author=Anvisa |author-link=Brazilian Health Regulatory Agency |date=2023-03-31 |title=RDC Nº 784 - Listas de Substâncias Entorpecentes, Psicotrópicas, Precursoras e Outras sob Controle Especial |trans-title=Collegiate Board Resolution No. 784 - Lists of Narcotic, Psychotropic, Precursor, and Other Substances under Special Control|url=https://www.in.gov.br/en/web/dou/-/resolucao-rdc-n-784-de-31-de-marco-de-2023-474904992 |url-status=live |archive-url=https://web.archive.org/web/20230803143925/https://www.in.gov.br/en/web/dou/-/resolucao-rdc-n-784-de-31-de-marco-de-2023-474904992 |archive-date=2023-08-03 |access-date=2023-08-16 |publisher=Diário Oficial da União |language=pt-BR |publication-date=2023-04-04}}

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| routes_of_administration = Suppository, injection

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| CAS_number_Ref = {{cascite|correct|??}}

| CAS_number = 63-12-7

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| ATC_prefix = none

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| IUPHAR_ligand = 7124

| DrugBank_Ref = {{drugbankcite|changed|drugbank}}

| DrugBank = DB00767

| ChemSpiderID_Ref = {{chemspidercite|changed|chemspider}}

| ChemSpiderID = 2252

| UNII_Ref = {{fdacite|correct|FDA}}

| UNII = 0475EA27Q3

| KEGG_Ref = {{keggcite|changed|kegg}}

| KEGG = D00243

| ChEMBL_Ref = {{ebicite|changed|EBI}}

| ChEMBL = 1201250

| synonyms =

| C=22 | H=32 | N=2 | O=5

| SMILES = CCN(CC)C(=O)C1CN2CCc3cc(OC)c(OC)cc3C2CC1OC(=O)C

| StdInChI_Ref = {{stdinchicite|changed|chemspider}}

| StdInChI = InChI=1S/C22H32N2O5/c1-6-23(7-2)22(26)17-13-24-9-8-15-10-20(27-4)21(28-5)11-16(15)18(24)12-19(17)29-14(3)25/h10-11,17-19H,6-9,12-13H2,1-5H3

| StdInChIKey_Ref = {{stdinchicite|changed|chemspider}}

| StdInChIKey = JSZILQVIPPROJI-UHFFFAOYSA-N

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Benzquinamide is a discontinued antiemetic drug used in post-operative care. It was first synthesised by Pfizer in the 1960s.{{cite journal|vauthors = Scriabine A, Weissman A, Finger KF|title=Benzquinamide|journal=JAMA|volume=184|issue=4|year=1963|pages=276–279|issn=0098-7484|doi=10.1001/jama.1963.73700170001010|pmid=13992595}}

{{cite journal | author = E.I. Goldenthal | journal = Toxicol. Appl. Pharmacol. | volume = 18 | pages = 185–207 | year = 1971 | doi = 10.1016/0041-008X(71)90328-0 | pmid = 5542824 | title = A compilation of LD50 values in newborn and adult animals | issue = 1| bibcode = 1971ToxAP..18..185G }}

References