N-Formylpiperidine

{{DISPLAYTITLE:N-Formylpiperidine}}

{{chembox

| Watchedfields = changed

| verifiedrevid = 419200108

| Name = N-Formylpiperidine

| ImageFile = N-Formylpiperidine.png

| ImageFile_Ref = {{chemboximage|correct|??}}

| ImageSize = 121

| ImageName = Skeletal formula of N-formylpiperidine

| PIN = Piperidine-1-carbaldehyde

| OtherNames = 1-Formylpiperidine

|Section1={{Chembox Identifiers

| CASNo_Ref = {{cascite|correct|??}}

| CASNo = 2591-86-8

| Beilstein = 107697

| PubChem = 17429

| ChemSpiderID = 16486

| ChemSpiderID_Ref = {{chemspidercite|correct|chemspider}}

| EINECS = 219-986-0

| DrugBank_Ref = {{drugbankcite|correct|drugbank}}

| DrugBank = DB04113

| MeSHName = N-Formylpiperidine

| RTECS = TN0380000

| UNNumber = 2810

| UNII_Ref = {{fdacite|correct|FDA}}

| UNII = ZIQ29H6CZG

| SMILES = O=CN1CCCCC1

| StdInChI = 1S/C6H11NO/c8-6-7-4-2-1-3-5-7/h6H,1-5H2

| StdInChI_Ref = {{stdinchicite|correct|chemspider}}

| InChI = 1/C6H11NO/c8-6-7-4-2-1-3-5-7/h6H,1-5H2

| StdInChIKey = FEWLNYSYJNLUOO-UHFFFAOYSA-N

| StdInChIKey_Ref = {{stdinchicite|correct|chemspider}}

| InChIKey = FEWLNYSYJNLUOO-UHFFFAOYAJ

}}

|Section2={{Chembox Properties

| C=6 | H=11 | N=1 | O=1

| Density = 1.019 g cm−3

| BoilingPtC = 222

| VaporPressure = 0.01 kPa

}}

|Section3={{Chembox Hazards

| GHSPictograms = {{GHS06}}{{GHS07}}

| GHSSignalWord = Danger

| HPhrases = {{H-phrases|302|311|315|319|335}}

| PPhrases = {{P-phrases|261|264|270|271|280|301+312|302+352|304+340|305+351+338|312|321|322|330|332+313|337+313|361|362|363|403+233|405|501}}

| NFPA-H = 2

| NFPA-F = 1

| NFPA-R = 0

| FlashPtC = 102

}}

}}

N-Formylpiperidine is an organic compound with the formula C6H11NO. It is the amide of formic acid and piperidine. It can be used as a polar aprotic solvent, with better hydrocarbon solubility than other amide solvents such as dimethylformamide (DMF).{{cite book |title=Kirk‑Othmer Encyclopedia of Chemical Technology |chapter=Pyridine and Pyridine Derivatives |author1=Eric F. V. Scriven |author2=Ramiah Murugan |year=2005 |name-list-style=amp |publisher=Wiley |doi=10.1002/0471238961.1625180919031809.a01.pub2|isbn=0471238961 }} It has also been used to transfer the formyl group to a Grignard reagent:{{OrgSynth | collvol = 7 | collvolpages = 451 | prep = cv7p0451 | title = Formyl Transfer to Grignard Reagents with N-Formylpiperidine: 3-Phenylpropionaldehyde | author = George Andrew Olah and Massoud Arvanaghi}}

: PhCH2CH2MgCl + C6H11NO → PhCH2CH2CHO

In some formylation reaction of alkyllithium compounds, N-formylpiperidine gives higher yields than the DMF.{{cite journal |author1=Lidija Bondarenko |author2=Ina Dix |author3=Heino Hinrichs |author4=Henning Hopf | title = Cyclophanes. Part LII:1 Ethynyl[2.2]paracyclophanes – New Building Blocks for Molecular Scaffolding | journal = Synthesis | volume = 2004| issue = 16 | pages = 2751–2759 | year = 2004 | doi = 10.1055/s-2004-834872}}

References

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{{DEFAULTSORT:Formylpiperidine, N-}}

Category:1-Piperidinyl compounds

Category:Formamides