ancestim

{{cs1 config|name-list-style=vanc}}

{{Drugbox

| Verifiedfields = changed

| verifiedrevid = 457130070

| IUPAC_name =

| image =

| tradename =

| Drugs.com = {{drugs.com|international|ancestim}}

| pregnancy_AU =

| pregnancy_US =

| pregnancy_category =

| legal_AU =

| legal_CA =

| legal_UK =

| legal_US =

| legal_status =

| routes_of_administration = s.c. injection only, premedication with H1 and H2 antihistamines and beta-receptor agonists for bronchodilation

| bioavailability =

| protein_bound =

| metabolism =

| elimination_half-life = 2.5 h

| excretion = renal: 90%

| ChemSpiderID_Ref = {{chemspidercite|changed|chemspider}}

| ChemSpiderID = none

| CAS_number_Ref = {{cascite|changed|??}}

| CAS_number = 163545-26-4

| ATC_prefix = L03

| ATC_suffix = AA12

| PubChem =

| DrugBank_Ref = {{drugbankcite|correct|drugbank}}

| DrugBank =

| UNII_Ref = {{fdacite|correct|FDA}}

| UNII = PYB4Q6JG41

| KEGG_Ref = {{keggcite|correct|kegg}}

| KEGG = D02937

| chemical_formula =

| molecular_weight =

}}

Ancestim is a recombinant methionyl human stem cell factor, branded by Amgen as StemGen. It was developed by Amgen and sold to Biovitrium, now Swedish Orphan Biovitrum, in December, 2008.Amgen press office. [http://www.amgen.com/media/biovitrum_amgen_deal.html Biovitrum Closes Product Acquisition Deal with Amgen] {{webarchive |url=https://web.archive.org/web/20120703015728/http://www.amgen.com/media/biovitrum_amgen_deal.html |date=July 3, 2012 }}

It is a 166 amino acid protein produced by E. coli bacteria into which a gene has been inserted for soluble human stem cell factor.{{cite journal |vauthors=da Silva MG, Pimentel P, Carvalhais A |title=Ancestim (recombinant human stem cell factor, SCF) in association with filgrastim does not enhance chemotherapy and/or growth factor-induced peripheral blood progenitor cell (PBPC) mobilization in patients with a prior insufficient PBPC collection |journal=Bone Marrow Transplant. |volume=34 |issue=8 |pages=683–91 |year=2004 |pmid=15322567 |doi=10.1038/sj.bmt.1704602|display-authors=etal|doi-access= |s2cid=21830065 }} It has a monomeric molecular weight of approximately 18,500 daltons and normally exists as a noncovalently associated dimer. The protein has an amino acid sequence that is identical to the natural sequence predicted from human DNA sequence analysis, except for the addition of an N-terminal methionine retained after expression in E. coli. Because Ancestim is produced in E. coli, it is nonglycosylated. Ancestim is supplied as a sterile, white, preservative-free, lyophilised powder for reconstitution and administration as a subcutaneous (SC) injection and is indicated for use in combination with filgrastim for mobilizing peripheral hematopoietic stem cells for later transplantation in certain cancer patients.{{cite web |url=http://www.sobi.com/en/Healthcare-Professionals/Products-alphabetical-list/Stemgen/ |title=Sobi's StemGen page |access-date=2013-12-30 |archive-url=https://web.archive.org/web/20160729205744/http://www.sobi.com/en/Healthcare-Professionals/Products-alphabetical-list/Stemgen/ |archive-date=2016-07-29 |url-status=dead }}

References

{{Growth factor receptor modulators}}

Category:Recombinant proteins

{{antineoplastic-drug-stub}}