batelapine
{{Short description|Chemical compound}}
{{One source|date=April 2021}}
{{Drugbox
| Verifiedfields =
| Watchedfields =
| verifiedrevid =
| IUPAC_name = 2-methyl-5-(4-methylpiperazin-1-yl)-11H-[1,2,4]triazolo[1,5-c][1,3]benzodiazepine
| image = Batelapine.svg
| width = 200
| tradename =
| routes_of_administration = By mouth
| bioavailability =
| metabolism =
| elimination_half-life = 8.1 Hours
| IUPHAR_ligand =
| CAS_number_Ref = {{cascite|correct|CAS}}
| CAS_number = 95634-82-5
| CAS_supplemental =
| ATC_prefix = None
| ATC_suffix =
| ATC_supplemental =
| PubChem = 60717
| DrugBank_Ref = {{drugbankcite|correct|drugbank}}
| DrugBank =
| ChemSpiderID_Ref = {{chemspidercite|changed|chemspider}}
| ChemSpiderID = 6721
| UNII_Ref = {{fdacite|changed|FDA}}
| UNII = P71TE299SG
| ChEMBL_Ref = {{ebicite|changed|EBI}}
| ChEMBL = 2110765
| KEGG_Ref = {{keggcite|changed|kegg}}
| KEGG =
| synonyms = CGS-13429
| C=16 | H=20 | N=6
| smiles = CC1=NN2C(=N1)CC3=CC=CC=C3N=C2N4CCN(CC4)C
| StdInChI_Ref = {{stdinchicite|correct|chemspider}}
| StdInChI = 1S/C16H20N6/c1-12-17-15-11-13-5-3-4-6-14(13)18-16(22(15)19-12)21-9-7-20(2)8-10-21/h3-6H,7-11H2,1-2H3
| StdInChIKey_Ref = {{stdinchicite|correct|chemspider}}
| StdInChIKey = PUHMYHQVPODHCZ-UHFFFAOYSA-N
}}
Batelapine (developmental code name CGS-13429) is a structural analogue of clozapine which was investigated as a potential antipsychotic.{{cite journal | vauthors = Chovan JP, Vermeulen JD | title = High-performance liquid chromatographic method for a clozapine analogue, CGS 13429, and its N-oxide and desmethyl metabolites | journal = Journal of Chromatography | volume = 494 | pages = 413–9 | date = September 1989 | pmid = 2573611 | doi = 10.1016/s0378-4347(00)82697-3 }}{{Cite web|url=https://adisinsight.springer.com/drugs/800007160|title=Batelapine - AdisInsight}}
References
{{Reflist}}
External links
- [https://adisinsight.springer.com/drugs/800007160 Batelapine - AdisInsight]
{{Tricyclics}}
Category:4-Methylpiperazin-1-yl compounds
Category:Triazolobenzodiazepines
{{Psychoactive-stub}}