clamoxyquine

{{Short description|Chemical compound}}

{{Drugbox

| IUPAC_name = 5-Chloro-7-({[3-(diethylamino)propyl]amino}methyl)quinolin-8-ol

| image = Clamoxyquine.svg

| tradename =

| pregnancy_category =

| legal_status =

| routes_of_administration =

| bioavailability =

| protein_bound =

| metabolism =

| elimination_half-life =

| excretion =

| CAS_number = 2545-39-3

| ATC_prefix = none

| ATC_suffix =

| PubChem = 18029

| DrugBank =

| ChEMBL = 2106065

| ChemSpiderID = 17033

| UNII_Ref = {{fdacite|correct|FDA}}

| UNII = JUN13FZ6RF

| C=17 | H=24 | Cl=1 | N=3 | O=1

| smiles = Clc1cc(c(O)c2ncccc12)CNCCCN(CC)CC

}}

Clamoxyquine (INN) or clamoxyquin (former BAN), as the pamoate or hydrochloride salt, is an antiamebic and antidiarrheal drug.

It has been used as a veterinary medicine to treat salmonids for infection with the myxozoan parasite Myxobolus cerebralis.

Synthesis

Antimalarial activity also predominates in a quinoline that bears a diaminoalkyl side chain at a rather different position from the other agents noted.

File:Clamoxyquin synthesis.svg

Thus, Mannich condensation of the hydroxyquinoline (1) with formaldehyde and N,N-diethylpropylenediamine affords clamoxyquin (2).

References

{{Reflist|2}}

Category:Veterinary drugs

Category:Quinolines

Category:Chloroarenes

Category:Diethylamino compounds

{{Antiinfective-drug-stub}}

{{Veterinary-med-stub}}