indisetron

{{Short description|Chemical compound}}

{{Infobox drug

| drug_name =

| INN =

| type =

| image = Indisetron.svg

| alt =

| caption =

| pronounce =

| tradename = Sinseron

| Drugs.com =

| MedlinePlus =

| pregnancy_AU =

| pregnancy_AU_comment =

| pregnancy_category=

| routes_of_administration =

| ATCvet =

| ATC_prefix = none

| ATC_suffix =

| legal_AU =

| legal_AU_comment =

| legal_BR =

| legal_BR_comment =

| legal_CA =

| legal_CA_comment =

| legal_DE =

| legal_DE_comment =

| legal_NZ =

| legal_NZ_comment =

| legal_UK =

| legal_UK_comment =

| legal_US =

| legal_US_comment =

| legal_EU =

| legal_EU_comment =

| legal_UN =

| legal_UN_comment =

| legal_status = Rx in Japan

| bioavailability =

| protein_bound =

| metabolism =

| metabolites =

| onset =

| elimination_half-life =

| duration_of_action=

| excretion =

| CAS_number = 141549-75-9

| PubChem = 178039

| DrugBank =

| UNII = 89RBZ66NVC

| ChEBI = 135344

| ChEMBL = 2104994

| ChemSpiderID = 2302029

| KEGG = D02632

| synonyms = N-3389

| smiles = CN1C[C@H]2CC(C[C@@H](C1)N2C)NC(=O)C3=NNC4=CC=CC=C43

| StdInChIKey = MHNNVDILNTUWNS-YHWZYXNKSA-N

| StdInChI = 1S/C17H23N5O/c1-21-9-12-7-11(8-13(10-21)22(12)2)18-17(23)16-14-5-3-4-6-15(14)19-20-16/h3-6,11-13H,7-10H2,1-2H3,(H,18,23)(H,19,20)/t11?,12-,13+

| IUPAC_name = N-[(1R,5S)-3,9-Dimethyl-3,9-diazabicyclo[3.3.1]nonan-7-yl]-1H-indazole-3-carboxamide

| C=17 | H=23 | N=5 | O=1

}}

Indisetron (INN; trade name Sinseron) is a drug used for prophylaxis of chemotherapy-induced nausea and vomiting. It was approved by Japan's Pharmaceuticals and Medical Devices Agency in 2004.

Indisetron exerts its effects as a dual serotonin 5-HT3 and 5-HT4 receptor antagonist.{{cite web | url = https://drugs.ncats.io/drug/89RBZ66NVC | title = Indisetron | work = Inxight: Drugs | publisher = National Center for Advancing Translational Sciences, National Institutes of Health }}{{cite journal | vauthors = Tsukagoshi S | title = [Introduction of novel anti-emetic agent, indisetron hydrochloride, developed recently in Japan] | language = Japanese | journal = Gan to Kagaku Ryoho. Cancer & Chemotherapy | volume = 32 | issue = 4 | pages = 567–73 | date = April 2005 | pmid = 15853230 | doi = | url = }}

See also

References

{{reflist}}

Category:Antiemetics

Category:Indazoles

Category:Amides

{{gastrointestinal-drug-stub}}