pentagestrone
{{short description|Chemical compound}}
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| IUPAC_name = 1-[(8R,9S,10R,13S,14S,17R)-3-cyclopentyloxy-17-hydroxy-10,13-dimethyl-1,2,7,8,9,11,12,14,15,16-decahydrocyclopenta[a]phenanthren-17-yl]ethanone
| image = Pentagestrone.svg
| width = 250px
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| class = Progestogen ether
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| CAS_number_Ref =
| CAS_number = 7001-56-1
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| PubChem = 3047827
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| ChemSpiderID_Ref =
| ChemSpiderID = 2310139
| UNII = L34YL185WL
| ChEMBL = 2104801
| synonyms = 17α-Hydroxyprogesterone 3-cyclopentyl enol ether
| C=26 | H=38 | O=3
| SMILES = CC(=O)C1(CCC2C1(CCC3C2CC=C4C3(CCC(=C4)OC5CCCC5)C)C)O
| StdInChI_Ref =
| StdInChI = 1S/C26H38O3/c1-17(27)26(28)15-12-23-21-9-8-18-16-20(29-19-6-4-5-7-19)10-13-24(18,2)22(21)11-14-25(23,26)3/h8,16,19,21-23,28H,4-7,9-15H2,1-3H3/t21-,22+,23+,24+,25+,26+/m1/s1
| StdInChIKey_Ref =
| StdInChIKey = RBFQPFFCDLXWQK-UXUCURBISA-N
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Pentagestrone ({{abbrlink|INN|International Nonproprietary Name}}), also known as 17α-hydroxyprogesterone 3-cyclopentyl enol ether, is a steroidal progestin of the 17α-hydroxyprogesterone group that was never marketed.{{cite book | vauthors = Elks J |title=The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies|url=https://books.google.com/books?id=0vXTBwAAQBAJ&pg=PA943|date=14 November 2014|publisher=Springer|isbn=978-1-4757-2085-3|pages=943–}}{{cite book| vauthors = Wermuth CG |title=The Practice of Medicinal Chemistry|url=https://books.google.com/books?id=Qmt1_DQkCpEC&pg=PA731|date=2 May 2011|publisher=Academic Press|isbn=978-0-08-056877-5|pages=731–|author-link=Camille Georges Wermuth}} An acetate ester, pentagestrone acetate (Gestovis, Gestovister), has been marketed for clinical use. Pentagestrone was described in the literature in 1960.
See also
References
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{{Progesterone receptor modulators}}
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