Cyprodenate
{{Short description|Chemical compound}}
{{Drugbox
| Watchedfields = changed
| verifiedrevid = 444141768
| IUPAC_name = 2-dimethylaminoethyl 3-cyclohexylpropanoate
| image = Cyprodenate.svg
| image_class = skin-invert-image
| width = 200
| tradename =
| Drugs.com = {{drugs.com|international|cyprodenate}}
| routes_of_administration =
| CAS_number_Ref = {{cascite|correct|??}}
| CAS_number = 15585-86-1
| ATC_prefix = N06BX04
| PubChem = 71875
| DrugBank_Ref = {{drugbankcite|correct|drugbank}}
| ChemSpiderID_Ref = {{chemspidercite|correct|chemspider}}
| ChemSpiderID = 64892
| ChEMBL = 2106590
| UNII_Ref = {{fdacite|correct|FDA}}
| UNII = I44VIC13P8
| KEGG_Ref = {{keggcite|correct|kegg}}
| KEGG = D07764
| C=13 | H=25 | N=1 | O=2
| smiles = CN(C)CCOC(=O)CCC1CCCCC1
| StdInChI_Ref = {{stdinchicite|correct|chemspider}}
| StdInChI = 1S/C13H25NO2/c1-14(2)10-11-16-13(15)9-8-12-6-4-3-5-7-12/h12H,3-11H2,1-2H3
| StdInChIKey_Ref = {{stdinchicite|correct|chemspider}}
| StdInChIKey = MPOYJPINNSIHAK-UHFFFAOYSA-N
}}
Cyprodenate (Actebral) is a stimulant drug.{{cite journal | vauthors = Dormard Y, Levron JC, Le Fur JM | title = Pharmacokinetic study of maleate acid of 2-(N,N-dimethylaminoethanol-14C1)-cyclohexylpropionate (cyprodenate) and of N,N-dimethylaminoethanol-14C1 in animals | journal = Arzneimittel-Forschung | volume = 25 | issue = 2 | pages = 201–7 | date = February 1975 | pmid = 1173033 }} It was used for counteracting the effects of benzodiazepine tranquillizer drugs before the development of newer antidotes such as flumazenil.{{cite journal | vauthors = Bobkov I, Morozov IS | title = [Correction of psychodepressive effects of benzodiazepine tranquilizers by administration of psychostimulants] | language = English | journal = Biulleten' Eksperimental'noi Biologii I Meditsiny | volume = 94 | issue = 10 | pages = 48–51 | date = October 1982 | pmid = 6129008 | doi = 10.1007/BF00827201 | s2cid = 19153614 }} It produces dimethylethanolamine as a metabolite.{{citation needed|date=September 2018}}
See also
References
{{Reflist}}
{{Stimulants}}
{{Acetylcholine receptor modulators}}
{{Monoamine releasing agents}}
Category:Dimethylamino compounds
{{nervous-system-drug-stub}}