Signaling peptide receptor
{{Short description|Cell surface receptors}}
Signaling peptide receptor is a type of receptor which binds one or more signaling peptides or signaling proteins.
An example is the tropomyosin receptor kinase B (TrkB), which is bound and activated by the neurotrophic protein brain-derived neurotrophic factor (BDNF). Another example is the μ-opioid receptor (MOR), which is bound and activated by the opioid peptide hormone β-endorphin.
Adiponectin receptor
{{Main|Adiponectin receptor}}
= AdipoR<sub>1</sub> =
{{Main|Adiponectin receptor 1}}
- Agonists
- Peptide
- Adiponectin
- ADP-355
- ADP-399
- Non-peptide
- AdipoRon
- (–)-Arctigenin
- Arctiin
- Gramine
- Matairesinol
- Antagonists
- Peptide
- ADP-400
= AdipoR<sub>2</sub> =
{{Main|Adiponectin receptor 2}}
- Agonists
- Peptide
- Adiponectin
- ADP-355
- ADP-399
- Non-peptide
- AdipoRon
- Deoxyschizandrin
- Parthenolide
- Syringing
- Taxifoliol
- Antagonists
- Peptide
- ADP-400
Angiotensin receptor
{{Main|Angiotensin receptor}}
Bradykinin receptor
{{Main|Bradykinin receptor}}
- Agonists
- Bradykinin
- Kallidin
- Antagonists
- FR-173657
- Icatibant
- LF22-0542
Cholecystokinin receptor
{{Main|Cholecystokinin receptor}}
= CCK<sub>A</sub> =
{{Main|Cholecystokinin A receptor}}
= CCK<sub>B</sub> =
{{Main|Cholecystokinin B receptor}}
= Unsorted =
- Antagonists
- Nastorazepide
Corticotropin-releasing hormone receptor
{{Main|Corticotropin-releasing hormone receptor}}
= CRF<sub>1</sub> =
{{Main|Corticotropin-releasing hormone receptor 1}}
= CRF<sub>2</sub> =
{{Main|Corticotropin-releasing hormone receptor 2}}
- Agonists
- Corticorelin
- Corticotropin-releasing hormone
- Sauvagine
- Urocortin
- Antagonists
- Astressin-B
Cytokine receptor
{{Main|Cytokine receptor}}
Endothelin receptor
{{Main|Endothelin receptor}}
Galanin receptor
{{Main|Galanin receptor}}
= GAL<sub>1</sub> =
{{Main|Galanin receptor 1}}
- Agonists
- Galanin
- Galanin (1-15)
- Galanin-like peptide
- Galmic
- Galnon
- NAX 810-2
- Antagonists
- C7
- Dithiepine-1,1,4,4-tetroxide
- Galantide (M15)
- M32
- M35
- M40
- SCH-202596
= GAL<sub>2</sub> =
{{Main|Galanin receptor 2}}
- Agonists
- Galanin
- Galanin (1-15)
- Galanin (2-11)
- Galanin-like peptide
- Galmic
- Galnon
- J18
- NAX 810-2
- Antagonists
- C7
- Galantide (M15)
- M32
- M35
- M40
- M871
= GAL<sub>3</sub> =
{{Main|Galanin receptor 3}}
- Agonists
- Galanin
- Galanin (1-15)
- Galmic
- Galnon
- Antagonists
- C7
- Galantide (M15)
- GalR3ant
- HT-2157
- M32
- M35
- M40
- SNAP-37889
- SNAP-398299
Growth hormone secretagogue receptor
{{Main|Growth hormone secretagogue receptor}}
Growth hormone receptor
{{Main|Growth hormone receptor}}
Growth-hormone-releasing hormone receptor
{{Main|Growth-hormone-releasing hormone receptor}}
Glucagon-like peptide receptor
= GLP-1 =
{{Main|Glucagon-like peptide-1 receptor}}
= GLP-2 =
{{Main|Glucagon-like peptide-2 receptor}}
- Agonists
- Apraglutide
- Elsiglutide
- Glepaglutide
- GLP-2
- Teduglutide
= Others =
- Propeptides
- Preproglucagon
- Proglucagon
Glucagon receptor
{{Main|Glucagon receptor}}
- Agonists
- Dasiglucagon
- Glucagon
- Oxyntomodulin
- Antagonists
- Adomeglivant
- L-168,049
- LGD-6972
- Propeptides
- Preproglucagon
- Proglucagon
Gonadotropin-releasing hormone receptor
{{Main|Gonadotropin-releasing hormone receptor}}
Gonadotropin receptor
{{Main|Gonadotropin receptor}}
Growth factor receptor
{{Main|Growth factor receptor}}
Insulin receptor
{{Main|Insulin receptor}}
- Agonists
- Chaetochromin (4548-G05)
- Insulin-like growth factor 1
- Insulin-like growth factor 2
- Insulin
- Insulin aspart
- Insulin degludec
- Insulin detemir
- Insulin glargine
- Insulin glulisine
- Insulin lispro
- Mecasermin
- Mecasermin rinfabate
- Antagonists
- BMS-754807
- S661
- S961
- Kinase inhibitors
- Linsitinib
- Antibodies
- Xentuzumab (against IGF-1 and IGF-2)
KiSS1-derived peptide receptor
{{Main|KiSS1-derived peptide receptor}}
Leptin receptor
{{Main|Leptin receptor}}
- Agonists
- Leptin
- Metreleptin
Melanin-concentrating hormone receptor
{{Main|Melanin-concentrating hormone receptor}}
= MCH<sub>1</sub> =
{{Main|Melanin-concentrating hormone receptor 1}}
- Agonists
- Melanin-concentrating hormone
- Antagonists
- ATC-0065
- ATC-0175
- GW-803430
- NGD-4715
- SNAP-7941
- SNAP-94847
= MCH<sub>2</sub> =
{{Main|Melanin-concentrating hormone receptor 2}}
- Agonists
- Melanin-concentrating hormone
Melanocortin receptor
{{Main|Melanocortin receptor}}
Neuropeptide FF receptor
{{Main|Neuropeptide FF receptor}}
- Agonists
- Neuropeptide AF
- Neuropeptide FF
- Neuropeptide SF (RFRP-1)
- Neuropeptide VF (RFRP-3)
- Antagonists
- BIBP-3226
- RF9
Neuropeptide S receptor
{{Main|Neuropeptide S receptor}}
- Agonists
- Neuropeptide S
- Antagonists
- ML-154
- SHA-68
Neuropeptide Y receptor
{{Main|Neuropeptide Y receptor}}
= Y<sub>1</sub> =
{{Main|Neuropeptide Y receptor Y1}}
- Agonists
- Neuropeptide Y
- Peptide YY
- Antagonists
- BIBO-3304
- BIBP-3226
- BVD-10
- GR-231118
- PD-160170
= Y<sub>2</sub> =
{{Main|Neuropeptide Y receptor Y2}}
= Y<sub>4</sub> =
- Agonists
- GR-231118
- Neuropeptide Y
- Pancreatic polypeptide
- Peptide YY
- Antagonists
- UR-AK49
= Y<sub>5</sub> =
{{Main|Neuropeptide Y receptor Y5}}
- Agonists
- BWX-46
- Neuropeptide Y
- Peptide YY
- Antagonists
- CGP-71683
- FMS-586
- L-152,804
- Lu AA-33810
- MK-0557
- NTNCB
- Velneperit (S-2367)
Neurotensin receptor
{{Main|Neurotensin receptor}}
= NTS<sub>1</sub> =
{{Main|Neurotensin receptor 1}}
- Agonists
- Neurotensin
- Neuromedin N
- Antagonists
- Meclinertant
- SR-142948
= NTS<sub>2</sub> =
{{Main|Neurotensin receptor 2}}
- Agonists
- Neurotensin
- Antagonists
- Levocabastine
- SR-142948
Opioid receptor
{{Main|Opioid receptor}}
Orexin receptor
{{Main|Orexin receptor}}
Oxytocin receptor
{{Main|Oxytocin receptor}}
Prolactin receptor
{{Main|Prolactin receptor}}
Parathyroid hormone receptor
{{Main|Parathyroid hormone receptor}}
Relaxin receptor
Somatostatin receptor
{{Main|Somatostatin receptor}}
Tachykinin receptor
{{Main|Tachykinin receptor}}
Thyrotropin-releasing hormone receptor
{{Main|Thyrotropin-releasing hormone receptor}}
Thyrotropin receptor
{{Main|Thyrotropin receptor}}
- Agonists
- Thyrotropin alfa
- TSH (thyrotropin)
Vasopressin receptor
{{Main|Vasopressin receptor}}
Vasoactive intestinal peptide receptor and Pituitary adenylate cyclase-activating peptide
{{Main|Vasopressin receptor}}
= VIPR<sub>1</sub> =
{{Main|VIPR1}}
- Agonists
- Peptide
- Bay 55-9837
- LBT-3393
- PACAP
- VIP
= VIPR<sub>2</sub> =
= PAC<sub>1</sub> =
{{Main|ADCYAP1R1}}
- Agonists
- PACAP
- PACAP (1-27)
- PACAP (1-38)
- Antagonists
- PACAP (6-38)
= Unsorted =
Others
- Endogenous
- Adrenomedullin
- Apelin
- Asprosin
- Bombesin
- Calcitonin
- Carnosine
- CART
- CLIP
- DSIP
- Enteroglucagon
- Formyl peptide
- GALP
- GIP
- GRP
- Integrin ligands
- collagens
- fibrinogen
- fibronectin
- laminins
- ICAM-1
- ICAM-2
- osteopontin
- VCAM-1
- vitronectin
- Kininogens
- Motilin
- Natriuretic peptides
- ANP
- BNP
- CNP
- urodilatin
- Nesfatin-1
- Neuromedin B
- Neuromedin N
- Neuromedin S
- Neuromedin U
- Obestatin
- Osteocalcin
- Resistin
- Secretin
- Thymopoietin
- Thymosins
- Thymulin
- Urotensin-II
- VGF
- Exogenous
- Lifitegrast (LFA-1 antagonist)
See also
References
{{reflist}}