List of combined sex-hormonal preparations#Androgens

{{Short description|None}}

This is a list of known combined sex-hormonal formulations. Brand names and developmental code names are in parentheses.

{{TOC limit|2}}

Androgens

=Injection=

==Marketed==

=Veterinary=

==Marketed==

Estrogens

=Oral=

==Marketed==

=Injection=

==Marketed==

==Never marketed==

Progestogens

=Injection=

==Marketed==

Androgens and estrogens

=Oral=

==Marketed==

=Injection=

==Marketed==

=Veterinary=

==Marketed==

Estrogens and progestogens

=Oral=

==Marketed==

In birth control pills:

  • Drospirenone/estetrol (Nextstellis, Drovelis, Lydisilka)
  • Estradiol/nomegestrol acetate (Naemis, Zoely)
  • Estradiol valerate/cyproterone acetate (Femilar)
  • Estradiol valerate/dienogest (Natazia, Qlaira)
  • Ethinylestradiol/chlormadinone acetate (Belara){{Cite web |url=https://www.ema.europa.eu/documents/psusa/chlormadinone-acetate/ethinylestradiol-list-nationally-authorised-medicinal-products-psusa/00000679/202111_en.pdf |title=Archived copy |access-date=2022-09-06 |archive-date=2022-09-06 |archive-url=https://web.archive.org/web/20220906054439/https://www.ema.europa.eu/en/documents/psusa/chlormadinone-acetate/ethinylestradiol-list-nationally-authorised-medicinal-products-psusa/00000679/202111_en.pdf |url-status=live }}
  • Ethinylestradiol/cyproterone acetate (Diane, Diane-35)
  • Ethinylestradiol/desogestrel (Alenvona, Apri,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=a9e08f9b-9862-4c2c-8302-53dc82d85126|title=Apri 28 Day- desogestrel and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=10 July 2021|archive-url=https://web.archive.org/web/20210710043751/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=a9e08f9b-9862-4c2c-8302-53dc82d85126|url-status=live}} Azurette,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=bff09a7b-aea6-460b-a263-44576e00f510|title=Azurette- desogestrel/ethinyl estradiol and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032434/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=bff09a7b-aea6-460b-a263-44576e00f510|url-status=live}} Bekyree,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=b9051bb5-21d0-4c76-9b70-c9cd89e67eb0|title=Bekyree- desogestrel and ethinyl estradiol and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032433/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=b9051bb5-21d0-4c76-9b70-c9cd89e67eb0|url-status=live}} Bimizza,{{cite web|url=https://www.medicines.org.uk/emc/product/9567/smpc|title=Bimizza 150 microgram/20 microgram Tablets - Summary of Product Characteristics (SmPC)|website=(emc)|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032432/https://www.medicines.org.uk/emc/product/9567/smpc|url-status=live}} Caziant,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=4e61bbb8-9b1b-4583-a7ad-1985b6d4de90|title=Caziant Triphasic Regimen- desogestrel and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032431/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=4e61bbb8-9b1b-4583-a7ad-1985b6d4de90|url-status=live}} Cesia,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=fed687f4-1ffa-49ec-92c9-4d09de17a833|title=Cesia- desogestrel and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032440/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=fed687f4-1ffa-49ec-92c9-4d09de17a833|url-status=live}} Cimizt,{{cite web|url=https://www.medicines.org.uk/emc/product/9568/smpc|title=Cimizt 150 microgram/30 microgram Tablets - Summary of Product Characteristics (SmPC)|website=(emc)|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032432/https://www.medicines.org.uk/emc/product/9568/smpc|url-status=live}} Cyclessa,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/archives/fdaDrugInfo.cfm?archiveid=311686|title=Cyclessa Tablets (desogestrel and ethinyl estradiol tablets USP)|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711034834/https://dailymed.nlm.nih.gov/dailymed/archives/fdaDrugInfo.cfm?archiveid=311686|url-status=live}} Cyred,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=2417aee4-6838-4ea6-8e0d-3144f522310c|title=Cyred EQ- desogestrel and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032437/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=2417aee4-6838-4ea6-8e0d-3144f522310c|url-status=live}} Denise, Desogen,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/archives/fdaDrugInfo.cfm?archiveid=276234|title=Desogen Tablets|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711034833/https://dailymed.nlm.nih.gov/dailymed/archives/fdaDrugInfo.cfm?archiveid=276234|url-status=live}} Desirett, Emoquette,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=ad604496-2df0-429e-b0da-12c6c38e61a5|title=Emoquette- desogestrel and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032436/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=ad604496-2df0-429e-b0da-12c6c38e61a5|url-status=live}} Enskyce,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=19dd4b23-b6e0-483a-97a7-fbabd201b1c2|title=Enskyce- desogestrel and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032438/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=19dd4b23-b6e0-483a-97a7-fbabd201b1c2|url-status=live}} Gedarel, Gracial, Isibloom,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=7dbc4cdf-4ce2-5c66-343f-df381f56692a|title=Isibloom- desogestrel and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032435/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=7dbc4cdf-4ce2-5c66-343f-df381f56692a|url-status=live}} Juleber,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=de9a2d1b-15f6-453f-b36b-1c2a43c4918d|title=Juleber- desogestrel and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032440/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=de9a2d1b-15f6-453f-b36b-1c2a43c4918d|url-status=live}} Kalliga, Kariva,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=7b11e11f-6977-4109-b9bd-a066e5d1278a|title=Kariva- desogestrel/ethinyl estradiol and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=10 July 2021|archive-url=https://web.archive.org/web/20210710043753/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=7b11e11f-6977-4109-b9bd-a066e5d1278a|url-status=live}} Kimidess,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/archives/fdaDrugInfo.cfm?archiveid=438314|title=Kimidess (Desogestrel and Ethinyl Estradiol Tablets, USP and Ethinyl Estradiol Tablets, USP), 0.15 mg/0.02 mg and 0.01 mg|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711034832/https://dailymed.nlm.nih.gov/dailymed/archives/fdaDrugInfo.cfm?archiveid=438314|url-status=live}} Laurina, Linessa, Marvelon,{{cite web|url=https://www.medicines.org.uk/emc/product/1359/smpc|title=Marvelon Tablets - Summary of Product Characteristics (SmPC)|website=(emc)|access-date=10 July 2021|archive-date=10 July 2021|archive-url=https://web.archive.org/web/20210710045255/https://www.medicines.org.uk/emc/product/1359/smpc|url-status=live}}{{cite web|url=https://tga-search.clients.funnelback.com/s/search.html?collection=tga-artg&profile=record&meta_i=42894|title=Marvelon desogestrel / ethinylestradiol 28 tablets|website=Therapeutic Goods Administration (TGA)|access-date=2021-07-11|archive-date=2021-07-11|archive-url=https://web.archive.org/web/20210711034319/https://tga-search.clients.funnelback.com/s/search.html?collection=tga-artg&profile=record&meta_i=42894|url-status=live}}{{cite web | title=Marvelon Product Information | website=Therapeutic Goods Administration (TGA) | url=https://www.ebs.tga.gov.au/ebs/picmi/picmirepository.nsf/pdf?OpenAgent&id=CP-2010-PI-06525-3 | access-date=10 July 2021 | archive-date=11 July 2021 | archive-url=https://web.archive.org/web/20210711034319/https://www.ebs.tga.gov.au/ebs/picmi/picmirepository.nsf/pdf?OpenAgent&id=CP-2010-PI-06525-3 | url-status=live }} Mercilon,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=7cb97fc9-59d2-3271-e053-2a91aa0afa5c|title=Mercilon- desogestrel, ethinyl estradiol tablet|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032439/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=7cb97fc9-59d2-3271-e053-2a91aa0afa5c|url-status=live}}{{cite web|url=https://www.medicines.org.uk/emc/product/1360/smpc|title=Mercilon Tablets - Summary of Product Characteristics (SmPC)|website=(emc)|access-date=10 July 2021|archive-date=10 July 2021|archive-url=https://web.archive.org/web/20210710043751/https://www.medicines.org.uk/emc/product/1360/smpc|url-status=live}} Mircette,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=a39bb616-9e84-4142-8450-824f88528906|title=Mircette- desogestrel/ethinyl estradiol and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=10 July 2021|archive-url=https://web.archive.org/web/20210710043752/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=a39bb616-9e84-4142-8450-824f88528906|url-status=live}} Mirvala, Novynette, Ortho-Cept,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/archives/fdaDrugInfo.cfm?archiveid=336921|title=Ortho-Cept Tablets (Desogestrel And Ethinyl Estradiol)|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711034836/https://dailymed.nlm.nih.gov/dailymed/archives/fdaDrugInfo.cfm?archiveid=336921|url-status=live}} Pimtrea,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=b716fd2a-b186-447a-85bd-6302284d14e5|title=Pimtrea- desogestrel/ethinyl estradiol and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032439/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=b716fd2a-b186-447a-85bd-6302284d14e5|url-status=live}} Reclipsen,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=a1e00bc6-7487-4057-9dcc-d0e2327d1d12|title=Reclipsen 28 Day- desogestrel and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032435/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=a1e00bc6-7487-4057-9dcc-d0e2327d1d12|url-status=live}} Regulon, Simliya,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=4161f614-6e55-4114-87f7-19bb77f6b09b|title=Simliya- desogestrel and ethinyl estradiol and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032434/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=4161f614-6e55-4114-87f7-19bb77f6b09b|url-status=live}} Solia, Velivet,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=a3ce5125-62ba-4983-93f0-91f254271605|title=Velivet Triphasic Regimen- desogestrel and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=10 July 2021|archive-url=https://web.archive.org/web/20210710043751/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=a3ce5125-62ba-4983-93f0-91f254271605|url-status=live}} Viorele,{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=39988aa6-8f68-40e8-9bdd-c40a3bdaad61|title=Viorele- desogestrel and ethinyl estradiol and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032437/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=39988aa6-8f68-40e8-9bdd-c40a3bdaad61|url-status=live}} Volnea{{cite web|url=https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=d7f3a118-4a1a-786e-c1db-01a0c2f2189d|title=Volnea- desogestrel and ethinyl estradiol kit|website=DailyMed|access-date=10 July 2021|archive-date=11 July 2021|archive-url=https://web.archive.org/web/20210711032434/https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=d7f3a118-4a1a-786e-c1db-01a0c2f2189d|url-status=live}})
  • Ethinylestradiol/dienogest (Valette)
  • Ethinylestradiol/dimethisterone (Oracon)
  • Ethinylestradiol/drospirenone (Yasmin, Yasminelle, Yaz)
  • Ethinylestradiol/drospirenone/levomefolic acid (Beyaz, Safyral)
  • Ethinylestradiol/etynodiol diacetate (Demulen)
  • Ethinylestradiol/gestodene (Femodene, Femodette, Gynera, Harmonet, Meliane, Minesse, Minulet)
  • Ethinylestradiol/levonorgestrel (Amethyst, Aviane, Balcoltra, Falmina, Levlen, Lillow, Orsythia, Vienva)
  • Ethinylestradiol/levonorgestrel/bisglycinate
  • Ethinylestradiol/levonorgestrel/ferrous fumarate
  • Ethinylestradiol/lynestrenol (Lyndiol)
  • Ethinylestradiol/medroxyprogesterone acetate (Gianda, Provest)
  • Ethinylestradiol/megestrol acetate (Nuvacon, Volidan)
  • Ethinylestradiol/norethisterone (Brevicon, Norinyl 1+35, Ortho-Novum 7/7/7, Taytulla, Tri-Norinyl, Zenchent)
  • Ethinylestradiol/norethisterone/ferrous fumarate (Blisovi 24 FE, Estrostep Fe, Femcon FE, Kaitlib FE, Lo Minastrin Fe, Loestrin 24 Fe, Microgestin 24 FE)
  • Ethinylestradiol/norethisterone acetate (FemHRT)
  • Ethinylestradiol/norethisterone acetate/ferrous fumarate
  • Ethinylestradiol/norgestimate (Ortho Tri-Cyclen, Sprintec)
  • Ethinylestradiol/norgestrel (Ovral)
  • Ethinylestradiol/norgestrienone (Miniplanor, Planor)
  • Ethinylestradiol/quingestanol acetate (Riglovis)
  • Ethinylestradiol sulfonate/norethisterone acetate (Deposiston)
  • Mestranol/anagestone acetate (Neo-Novum)
  • Mestranol/chlormadinone acetate (C-Quens, Lutedion)
  • Mestranol/etynodiol diacetate (Ovulen)
  • Mestranol/hydroxyprogesterone acetate (Hormolidin)
  • Mestranol/lynestrenol (Lyndiol)
  • Mestranol/norethisterone (Norethin, Noriday, Norinyl, Norquen, Ortho-Novum)
  • Mestranol/noretynodrel (Enavid, Enovid)
  • Quinestrol/etynodiol diacetate (Soluna)
  • Quinestrol/levonorgestrel (Yuèkětíng, Àiyuè)
  • Quinestrol/norgestrel (Compound Norgestrel)
  • Quinestrol/quingestanol acetate (Unovis)

For menopausal hormone therapy and/or gynecological disorders:

==Never or not yet marketed==

In birth control pills:

=Transdermal=

==Marketed==

=Vaginal=

==Marketed==

=Injection=

==Marketed==

==Never marketed==

=Veterinary=

==Marketed==

Androgens and progestogens

=Oral=

==Marketed==

=Injection=

==Marketed==

  • Testosterone propionate/progesterone (Testoluton){{cite book|author=Josef Kimmig|title=Therapie der Haut- und Geschlechtskrankheiten|url=https://books.google.com/books?id=txrUBgAAQBAJ&pg=PA508|date=14 March 2013|publisher=Springer-Verlag|isbn=978-3-642-94850-3|pages=508–|access-date=3 June 2019|archive-date=29 August 2021|archive-url=https://web.archive.org/web/20210829162439/https://books.google.com/books?id=txrUBgAAQBAJ&pg=PA508|url-status=live}}{{cite book|author1=Hans Hermann Julius Hager|author2=Walther Kern|author3=Paul Heinz List|author4=Hermann Josef Roth|title=Hagers Handbuch der Pharmazeutischen Praxis: Für Apotheker, Arzneimittelhersteller, Ärzte und Medizinalbeamte: Wirkstoffgruppen II Chemikalien und Drogen (A-AL)|url=https://books.google.com/books?id=a2a0BgAAQBAJ&pg=PA185|date=29 July 2013|publisher=Springer-Verlag|isbn=978-3-662-25655-8|pages=143, 185–187|access-date=3 June 2019|archive-date=6 September 2022|archive-url=https://web.archive.org/web/20220906054441/https://books.google.com/books?id=a2a0BgAAQBAJ&pg=PA185|url-status=live}}{{cite book|author1=Georg Arends|author2=Heinrich Zörnig|author3=Hermann Hager|author4=Georg Frerichs, Walther Kern|title=Hagers Handbuch der pharmazeutischen Praxis: Für Apotheker, Arzneimittelhersteller, Drogisten, Ärzte u. Medizinalbeamte|url=https://books.google.com/books?id=8bLwBgAAQBAJ&pg=PA1163|date=14 December 2013|publisher=Springer-Verlag|isbn=978-3-662-36329-4|pages=1163–1164|access-date=3 June 2019|archive-date=6 September 2022|archive-url=https://web.archive.org/web/20220906054441/https://books.google.com/books?id=8bLwBgAAQBAJ&pg=PA1163|url-status=live}}{{cite journal|title=Spezialitäten|journal=Klinische Wochenschrift|volume=30|issue=15–16|year=1952|pages=367|issn=0023-2173|doi=10.1007/BF01472052|s2cid=264011779 }}[https://www.jstage.jst.go.jp/article/sanpunosinpo1949/8/2/8_2_100/_pdf Archived copy] {{Webarchive|url=https://web.archive.org/web/20190609083210/https://www.jstage.jst.go.jp/article/sanpunosinpo1949/8/2/8_2_100/_pdf |date=2019-06-09 }}

=Veterinary=

==Marketed==

Estrogens, progestogens, and androgens

=Oral=

==Marketed==

==Not yet marketed==

=Sublingual=

==Marketed==

=Injection=

==Marketed==

==Never marketed==

=Veterinary=

==Marketed==

Miscellaneous

=Oral=

==Marketed==

==Never marketed==

=Transdermal=

==Marketed==

=Vaginal=

==Marketed==

=Mixed=

==Marketed==

See also

References

{{Reflist}}

{{Androgens and antiandrogens}}

{{Estrogens and antiestrogens}}

{{Progestogens and antiprogestogens}}

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Category:Anabolic–androgenic steroids

Sex-hormonal preparations

Category:Drug-related lists

Category:Estrogens

Category:Progestogens